Enzyme source
Km
Vmax
CLint
CLint fold (CYP2J2 / CYPs)
HLM 22.81 ± 2.370 91.28 ± 3.233 4.002
CYP2J2 19.37 ± 1.932 753.9 ± 19.97 38.92
CYP3A4 46.98 ± 4.800 47.24 ± 1.843 1.006 38.68
CYP2D6 98.78 ± 8.839 59.94 ± 2.597 0.607 64.11
CYP4F3 75.19 ± 5.312 29.42 ± 0.898 0.391 99.54