Dose
Median Cmax (µg/mL)
Median tmax (hours)
AUC(0-last) (µg.h/mL)
t1/2 λz (h)
Single 2.00 mg.kg-1 45.1 1.5 1180 37.7
Single 4.00 mg.kg-1 77.7 0.75 2373 44.3
Repeated 4.00 mg.kg-1, Day 1 85.7 0.5 1810 N/A
Repeated 4.00 mg.kg-1, Day 2 113.1 1 2570 N/A
Repeated 4.00 mg.kg-1, Day 3 149 2 7040 74.4