parameter |
Fasting |
Fasting |
Fed |
Fed |
|
R(N(R1)=48,N(R2)=46) |
T(N(T1)=48,N(T2)=47) |
R(N=48) |
T(N=48) |
Cmax, ng/mL |
26.1±12.1 |
29.5±13.1 |
29.9±10.8 |
32.7±12.4 |
Tmax, h |
24.00 (4.00,36.00) |
24.00(4.00,48.00) |
6.00
(4.00,24.00) |
7.00(4.00,48.00) |
AUC0-t,ng∙h/mL |
686.14±372.05 |
744.92±410.67 |
657.35±340.71 |
736.89±368.76 |
AUC0-∞ ,ng∙h/mL |
695.00±388.67 |
772.99±426.05 |
673.95±349.94 |
732.46±358.32 |
t1/2, h |
7.93±3.01 |
7.12±2.65 |
7.22±3.06 |
6.57±2.12 |