Company
|
Sankyo
|
Merck
|
Merck
|
Sankyo
|
Sandoz
|
Pfizer
|
AstraZeneca
|
JINGXIN
|
Half-life
|
/
|
3 h
|
2-3 h
|
1.5 h
|
2.3±0.9 h
|
14 h
|
19 h
|
11 h
|
Clearance
|
/
|
Hepatic
|
Hepatic
|
Hepatic and renal
|
Hepatic
|
Hepatic
|
Hepatic and renal
|
Hepatic
|
Form Administered
|
/
|
Inactive lactone
|
Inactive lactone
|
Active hydroxy acid
|
Active hydroxy acid
|
Active hydroxy acid
|
Active hydroxy acid
|
Active hydroxy acid
|
Solubility
|
/
|
Lipophilic
|
Lipophilic
|
Hydrophilic
|
Lipophilic
|
Lipophilic
|
Hydrophilic
|
Lipophilic
|
Derivative
|
Fungal
|
Fungal
|
Fungal
|
Fungal
|
Synthetic
|
Synthetic
|
Synthetic
|
Synthetic
|
Structure
|
|
|
|
|
|
|
|
|
Generation
|
/
|
First
|
First
|
Second
|
Second
|
Third
|
Third
|
Third
|
Drug name
|
Compactin
|
Lovastatin
|
Simvastatin
|
Pravastatin
|
Fluvastatin
|
Atorvastatin
|
Rosuvastatin
|
Pitavastatin
|